SCHEMBL7225460

SCHEMBL7225460

Cc1ccn(-c2ccc(C(=O)N3Cc4nnnn4Cc4ccccc43)c(Cl)c2)n1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 20/20 0.68
AVPR1A P37288 11/20 0.68
OXTR P30559 3/20 0.68
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6623456 0.83 AVPR2 (0.77) AVPR2AVPR1AOXTR
SCHEMBL6627050 0.81 AVPR2 (1.00) AVPR2AVPR1AOXTR
SCHEMBL6623504 0.80 AVPR2 (0.76) AVPR2AVPR1AOXTRCYP3A4CYP2C19
SCHEMBL6624422 0.79 AVPR2 (0.73) AVPR2AVPR1AOXTRCYP3A4CYP2C19
SCHEMBL6624625 0.76 AVPR2 (0.68) AVPR2AVPR1AOXTR
SCHEMBL14130377 0.75 AVPR2 (0.66) AVPR2AVPR1AOXTRCYP3A4CYP2C19
SCHEMBL6618394 0.74 AVPR2 (0.71) AVPR2AVPR1AOXTRCYP3A4CYP2C19
SCHEMBL6615751 0.74 AVPR2 (1.00) AVPR2AVPR1AOXTRCYP3A4CYP2C19
SCHEMBL17158263 0.74 AVPR2 (0.69) AVPR2AVPR1AOXTRCYP3A4CYP2C19
SCHEMBL14130132 0.73 AVPR2 (0.60) AVPR2AVPR1AOXTRCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6511974-B1 Non-peptidic and have good oral bioavailability, specific vasopressin V2 agonists, therefore do not raise blood pressure WYETH 2003-01-28 US claimed
US-6511974-B1 Non-peptidic and have good oral bioavailability, specific vasopressin V2 agonists, therefore do not raise blood pressure WYETH 2003-01-28 US disclosed