SCHEMBL7230894

SCHEMBL7230894

C/C=C(\CN1CCNCC1)CN1CCNC1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 2/20 0.41
CHRM3 P20309 2/20 0.41
SIGMAR1 Q99720 6/20 0.38
SMN1; SMN2 Q16637 3/20 0.32
ALDH1A1 P00352 1/20 0.32
STAT6 P42226 1/20 0.32
HSD17B10 Q99714 1/20 0.32
POLB P06746 1/20 0.31
CXCR4 P61073 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230900 1.00 CHRM5 (0.41) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7221968 0.96 CHRM5 (0.35) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7228712 0.92 CHRM5 (0.46) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7229670 0.91 CHRM5 (0.38) CHRM5CHRM3SIGMAR1ALDH1A1POLB
SCHEMBL7229675 0.91 CHRM5 (0.38) CHRM5CHRM3SIGMAR1ALDH1A1POLB
SCHEMBL7223188 0.88 KDM4E (0.38) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7223190 0.88 KDM4E (0.38) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7223180 0.88 KDM4E (0.38) CHRM5CHRM3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL7708079 0.86 CHRM5 (0.33) CHRM5CHRM3SIGMAR1
SCHEMBL7710764 0.86 CHRM5 (0.33) CHRM5CHRM3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6552226-B1 Rapid; low temperature; one pot synthesis; reduced catalytic quantities of such as lewis acid and tertiary amine; entiomerically pure products THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2003-04-22 US disclosed
WO-2002026683-A1 TANDEM ACYL-CLAISEN REARRANGEMENT IN THE PREPARATION OF CHIRAL PRODUCTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2002-04-04 WO disclosed