SCHEMBL7233641

SCHEMBL7233641

COCCNCc1ccc2nc3sc(C(=O)N(C)c4ccccc4)cn3c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 3/20 0.51
HPGD P15428 2/20 0.36
RAB9A P51151 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
AVPR1B P47901 1/20 0.36
ITK Q08881 1/20 0.35
LMNA P02545 2/20 0.35
ACSS2 Q9NR19 1/20 0.35
METTL3 Q86U44 1/20 0.34
HDAC1 Q13547 2/20 0.34
NPC1 O15118 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
SLC40A1 Q9NP59 1/20 0.34
TP53 P04637 1/20 0.34
CHEK1 O14757 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7233455 0.99 GRM1 (0.50) GRM1HPGDRAB9ACYP1A2CYP2C9
SCHEMBL658903 0.85 GRM1 (0.69) GRM1HPGDRAB9ALMNANPC1
SCHEMBL7241303 0.85 GRM1 (0.51) GRM1HPGDRAB9ACYP1A2CYP2C9
Hydrochloric Acid SCHEMBL7241479 0.84 GRM1 (0.51) GRM1HPGDRAB9ACYP1A2CYP2C9
Hydrochloric Acid SCHEMBL7240261 0.82 GRM1 (0.47) GRM1HPGDRAB9ALMNANPC1
SCHEMBL7233634 0.82 GRM1 (0.75) GRM1HPGDAVPR1BITKLMNA
Hydrochloric Acid SCHEMBL7233449 0.81 GRM1 (0.74) GRM1HPGDAVPR1BITKLMNA
Hydrochloric Acid SCHEMBL7233122 0.81 GRM1 (0.46) GRM1HPGDRAB9ALMNANPC1
SCHEMBL4693193 0.80 GRM1 (0.46) GRM1HPGDRAB9ACYP1A2CYP2C9
SCHEMBL7233822 0.80 GRM1 (0.50) GRM1RAB9AITKLMNAACSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6642264-B1 Thiazolo(3,2-a)benzoimidazole derivatives act specifically on metabotropic glutamate receptors and are used as medicaments. YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2003-11-04 US claimed
EP-1167369-A1 NOVEL THIAZOLOBENZIMIDAZOLE DERIVATIVES YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2002-01-02 EP claimed
US-6642264-B1 Thiazolo(3,2-a)benzoimidazole derivatives act specifically on metabotropic glutamate receptors and are used as medicaments. YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2003-11-04 US disclosed
EP-1167369-A1 NOVEL THIAZOLOBENZIMIDAZOLE DERIVATIVES YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2002-01-02 EP disclosed