SCHEMBL7241122

SCHEMBL7241122

COc1ccc2c(c1)-c1nc(Nc3cc(OC)c(OC)c(OC)c3)ncc1CC2(C)C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 3/20 0.65
KDR P35968 12/20 0.55
PLK1 P53350 10/20 0.49
IGF1R P08069 3/20 0.47
AURKA O14965 1/20 0.47
DAPK3 O43293 1/20 0.47
JAK2 O60674 1/20 0.47
PAK4 O96013 1/20 0.47
ABL1 P00519 1/20 0.47
NTRK1 P04629 1/20 0.47
LCK P06239 1/20 0.47
CSF1R P07333 1/20 0.47
RET P07949 1/20 0.47
MET P08581 1/20 0.47
PDGFRB P09619 1/20 0.47
FGFR1 P11362 1/20 0.47
PDGFRA P16234 1/20 0.47
PRKACA P17612 1/20 0.47
FLT1 P17948 1/20 0.47
LTK P29376 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7242637 0.94 FYN (0.59) FYNKDRPLK1IGF1RAURKA
SCHEMBL7234789 0.89 KDR (0.64) FYNKDRPLK1IGF1RJAK2
Hydrochloric Acid SCHEMBL7240520 0.88 FYN (0.56) FYNKDRPLK1IGF1RAURKA
SCHEMBL7240926 0.88 FYN (0.57) FYNKDRPLK1IGF1RIKBKB
Hydrochloric Acid SCHEMBL7240228 0.88 FYN (0.65) FYNKDRPLK1IGF1RPTK2
SCHEMBL7232580 0.86 KDR (0.63) FYNKDRPLK1IGF1RAURKA
SCHEMBL7231388 0.86 FYN (0.61) FYNKDRPLK1IGF1RIKBKB
Hydrochloric Acid SCHEMBL7232574 0.85 PLK1 (0.64) FYNKDRPLK1IGF1RPTK2
SCHEMBL7001153 0.85 FYN (0.56) FYNKDRPLK1IGF1RIKBKB
SCHEMBL7237418 0.85 FYN (0.65) FYNKDRPLK1IGF1RAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6599908-B1 Potent and selective inhibitors of the protein tyrosine kinases p56lck and p59fyn CELLTECH R & D LIMITED (GB) 2003-07-29 US disclosed
US-6057329-A Fused polycyclic 2-aminopyrimidine derivatives CELLTECH THERAPEUTICS LIMITED (GB) 2000-05-02 US disclosed