SCHEMBL7243277

SCHEMBL7243277

CCN(CC)CCOc1c(OC)cc(Nc2ncc3c(n2)-c2cc(OC)cnc2CC3)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FYN P06241 3/20 0.54
KDR P35968 6/20 0.42
RIPK2 O43353 1/20 0.41
NOD2 Q9HC29 1/20 0.41
IKBKB O14920 1/20 0.41
PDGFRB P09619 2/20 0.40
IGF1R P08069 4/20 0.39
PLK1 P53350 3/20 0.38
CCNA2 P20248 2/20 0.37
CDK2 P24941 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230375 0.88 FYN (0.51) FYNKDRIKBKBPDGFRBIGF1R
SCHEMBL7241210 0.87 FYN (0.49) FYNKDRIKBKBPDGFRBIGF1R
SCHEMBL7240933 0.85 FYN (0.52) FYNKDRRIPK2NOD2IKBKB
SCHEMBL7240926 0.80 FYN (0.57) FYNKDRRIPK2NOD2IKBKB
SCHEMBL7234420 0.80 IKBKB (0.48) FYNKDRIKBKBIGF1RPLK1
SCHEMBL7002121 0.77 FYN (0.66) FYNKDRIKBKBIGF1RPLK1
Hydrochloric Acid SCHEMBL7240520 0.75 FYN (0.56) FYNKDRRIPK2NOD2IKBKB
SCHEMBL7237418 0.73 FYN (0.65) FYNKDRIKBKBPDGFRBIGF1R
SCHEMBL7230505 0.73 FYN (0.49) FYNKDRIKBKBPDGFRBIGF1R
SCHEMBL7234843 0.72 FYN (0.58) FYNKDRIKBKBPDGFRBIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6599908-B1 Potent and selective inhibitors of the protein tyrosine kinases p56lck and p59fyn CELLTECH R & D LIMITED (GB) 2003-07-29 US disclosed
US-6057329-A Fused polycyclic 2-aminopyrimidine derivatives CELLTECH THERAPEUTICS LIMITED (GB) 2000-05-02 US disclosed