SCHEMBL7253295

SCHEMBL7253295

N#Cc1ccc2cc1Oc1ccc3cccc(c3c1)N1CCN(CC1=O)C(=O)c1cnc3n1C2CC3

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FNTA P49354 18/20 0.51
PGGT1B P53609 17/20 0.51
FNTB P49356 15/20 0.51
DNAJA1 P31689 1/20 0.51
KCNH2 Q12809 9/20 0.49
CYP3A4 P08684 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7252683 0.99 FNTA (0.51) FNTAPGGT1BFNTBDNAJA1KCNH2
SCHEMBL7248216 0.82 FNTA (0.51) FNTAPGGT1BFNTBDNAJA1KCNH2
SCHEMBL7252273 0.82 FNTA (0.51) FNTAPGGT1BFNTBDNAJA1KCNH2
Hydrochloric Acid SCHEMBL7247014 0.81 FNTA (0.50) FNTAPGGT1BFNTBDNAJA1KCNH2
Hydrochloric Acid SCHEMBL7253913 0.81 FNTA (0.50) FNTAPGGT1BFNTBDNAJA1KCNH2
Hydrochloric Acid SCHEMBL7248127 0.81 FNTA (0.50) FNTAPGGT1BFNTBDNAJA1KCNH2
SCHEMBL7184432 0.77 FNTA (0.51) FNTAPGGT1BFNTBDNAJA1KCNH2
SCHEMBL7181655 0.77 FNTA (0.51) FNTAPGGT1BFNTBDNAJA1KCNH2
SCHEMBL7184844 0.77 FNTA (0.51) FNTAPGGT1BFNTBDNAJA1KCNH2
SCHEMBL7185080 0.77 FNTA (0.51) FNTAPGGT1BFNTBDNAJA1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6534506-B2 For therapy of cancer, neurofibromin benign proliferative disorder; blindness related to retinal vascularization; infections from hepatitis delta and related viruses; prophylaxis of restenosis; polycystic kidney disease MERCK & CO., INC. 2003-03-18 US claimed
US-20020123497-A1 Inhibitors of prenyl-protein transferase MERCK SHARP & DOHME CORP. 2002-09-05 US claimed
WO-2001077116-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-10-18 WO claimed
US-6534506-B2 For therapy of cancer, neurofibromin benign proliferative disorder; blindness related to retinal vascularization; infections from hepatitis delta and related viruses; prophylaxis of restenosis; polycystic kidney disease MERCK & CO., INC. 2003-03-18 US disclosed
US-20020123497-A1 Inhibitors of prenyl-protein transferase MERCK SHARP & DOHME CORP. 2002-09-05 US disclosed
WO-2001077116-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020123497-A1 Inhibitors of prenyl-protein transferase FNTA, KRAS, NRAS FNTA 1/4885PGGT1B 122/4885FNTB 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.