SCHEMBL7258367

SCHEMBL7258367

O=c1[nH]c2ncc(-c3ccncc3)cc2c(=O)n1CC(S)CS

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
GRIN1 Q05586 13/20 0.40
GRIN2B Q13224 13/20 0.40
CHEK1 O14757 2/20 0.39
METAP2 P50579 2/20 0.37
AXL P30530 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7100335 1.00 PDE3B (0.41) PDE3BPDE3AGRIN1GRIN2BCHEK1
SCHEMBL7019405 0.77 FEN1 (0.56)
SCHEMBL7019409 0.77 FEN1 (0.56)
SCHEMBL7014592 0.71 FEN1 (0.35)
SCHEMBL7014590 0.71 FEN1 (0.35)
SCHEMBL7020404 0.71 KDM4E (0.45)
SCHEMBL7020408 0.71 KDM4E (0.45)
SCHEMBL7022651 0.70
SCHEMBL7022655 0.70
SCHEMBL11236623 0.69 GRIN1 (0.55) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003089416-A1 SUBSTITUTED PYRIMIDINE-2,4(1H,3H)-DIONES FOR USE AS MATRIX METALLOPROTEINASE (MMP) INHIBITORS IBFB GMBH (DE) 2003-10-30 WO disclosed