SCHEMBL7259642

SCHEMBL7259642

CCOc1c(N[C@@H](Cc2ccc(Nc3nc(C)cc4ccncc34)cc2)C(=O)O)c(=O)c1=O

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.40
ITGA4 P13612 19/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7259650 1.00 ITGB1 (0.40) ITGB1ITGA4MAPT
SCHEMBL7264625 0.90 ITGB1 (0.43) ITGB1ITGA4
SCHEMBL7264618 0.90 ITGB1 (0.43) ITGB1ITGA4
SCHEMBL7264734 0.90 ITGB1 (0.43) ITGB1ITGA4MAPT
SCHEMBL7264754 0.90 ITGB1 (0.43) ITGB1ITGA4MAPT
SCHEMBL7259942 0.85 ITGB1 (0.55) ITGB1ITGA4
SCHEMBL7264635 0.85 ITGB1 (0.47) ITGB1ITGA4
SCHEMBL7264644 0.85 ITGB1 (0.47) ITGB1ITGA4
SCHEMBL7259595 0.84 ITGB1 (0.51) ITGB1ITGA4
SCHEMBL7259040 0.84 POLB (0.40) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545013-B2 Of squaric acids; inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders or disorders involving the inappropriate growth or migration of cells. CELLTECH R&D LIMITED (GB) 2003-04-08 US disclosed