SCHEMBL7260702

SCHEMBL7260702

CC(C)c1[nH]nc2c(NCc3c(O)cc(Cl)cc3O)nc(NCC(O)C(C)C)nc12

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 16/20 0.52
CCNE1 P24864 14/20 0.52
CDK5 Q00535 13/20 0.48
CDK1 P06493 7/20 0.48
CDK9 P50750 3/20 0.48
CDK7 P50613 2/20 0.48
CDK5R1 Q15078 3/20 0.43
CCNT1 O60563 2/20 0.43
CCNH P51946 1/20 0.43
AURKA O14965 1/20 0.41
CCNE2 O96020 1/20 0.41
CCNB1 P14635 6/20 0.40
CDK4 P11802 2/20 0.40
CCNA2 P20248 2/20 0.40
CCND1 P24385 2/20 0.40
CDK6 Q00534 1/20 0.40
CCNB2 O95067 4/20 0.39
CCNB3 Q8WWL7 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7259669 0.85 CDK2 (0.55) CDK2CCNE1CDK5CDK1CDK9
SCHEMBL2908707 0.83 CDK2 (0.52) CDK2CCNE1CDK5CDK1CDK9
SCHEMBL2908697 0.83 CDK2 (0.52) CDK2CCNE1CDK5CDK1CDK9
SCHEMBL3794926 0.76 CDK2 (0.52) CDK2CCNE1CDK5CDK1CDK9
SCHEMBL3444052 0.73 CDK2 (0.39) CDK2CCNE1CDK5CDK1CDK9
SCHEMBL3717049 0.71 CDK2 (0.50) CDK2CCNE1CDK5CDK1CDK9
SCHEMBL3444820 0.71 BCDIN3D (0.35) CDK2CCNE1CDK5CDK9CDK7
SCHEMBL3444444 0.70 CDK2 (0.42) CDK2CCNE1CDK5CDK1CDK9
SCHEMBL3724482 0.70 CDK2 (0.51) CDK2CCNE1CDK5CDK1CDK9
SCHEMBL3722157 0.69 CDK2 (0.57) CDK2CCNE1CDK5CDK1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003082872-A1 NOVEL PYRAZOLO[4,3-D]PYRIMIDINES, PROCESSES FOR THEIR PREPARATION AND METHODS FOR THERAPY USTAV EXPERIMENTALNI BOTANIKY AV CR (INSTITUTE OF EXPERIMENTAL BOTANY ACADEMY OF SCIENCES OF THE CZECH REPUBLIC) (CZ) 2003-10-09 WO disclosed