SCHEMBL7263122

SCHEMBL7263122

O=C1CNC(=O)N1Cc1ccc(I)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.69
GSK3B P49841 1/20 0.69
KMT2A Q03164 6/20 0.53
MEN1 O00255 5/20 0.53
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
ALDH1A1 P00352 3/20 0.42
TSHR P16473 1/20 0.42
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
FAAH O00519 1/20 0.39
MGLL Q99685 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
HTR2C P28335 1/20 0.38
GRM2 Q14416 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6293317 0.84 KMT2A (0.73) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL8320050 0.82 SMN1; SMN2 (0.73) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL29234520 0.82 GSK3A (0.69) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL5311390 0.82 GSK3A (0.69) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL3318940 0.81 GSK3A (1.00) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL5182321 0.80 GSK3A (0.66) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL30953279 0.80 GSK3A (0.71) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL378362 0.79 GSK3A (0.65) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL4455461 0.79 GSK3A (0.69) GSK3AGSK3BKMT2AMEN1GAA
SCHEMBL7267266 0.78 GSK3A (0.63) GSK3AGSK3BKMT2AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667334-B1 Inhibitors of adhesion and migration of leukocytes and/or antagonists of adhesion receptor VLA-4 belonging to integrins group AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-12-23 US disclosed