SCHEMBL7267686

SCHEMBL7267686

Cc1ccn2cc(C(=O)O)nc2c1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.53
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
KDM4E B2RXH2 7/20 0.35
POLB P06746 2/20 0.35
TDP1 Q9NUW8 3/20 0.34
TSHR P16473 2/20 0.34
ALOX15 P16050 1/20 0.34
ACMSD Q8TDX5 1/20 0.34
RAB9A P51151 3/20 0.34
ALDH1A1 P00352 2/20 0.34
NPC1 O15118 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
DHODH Q02127 1/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8378456 0.84 RXFP1 (0.50) RXFP1PTGS1PTGS2KDM4EPOLB
SCHEMBL7268780 0.80 KDM4E (0.59) RXFP1KDM4EPOLBRAB9AALDH1A1
SCHEMBL1758978 0.80 RXFP1 (0.56) RXFP1PTGS1PTGS2KDM4EPOLB
SCHEMBL3305733 0.71 PTGS1 (0.56) RXFP1PTGS1PTGS2KDM4EPOLB
SCHEMBL23571486 0.71 PTGS1 (0.47) RXFP1PTGS1PTGS2KDM4EPOLB
SCHEMBL2505187 0.71 PTGS1 (0.51) RXFP1PTGS1PTGS2KDM4ETDP1
SCHEMBL26922447 0.71 PTGS1 (0.44) RXFP1PTGS1PTGS2KDM4ETDP1
SCHEMBL19660422 0.70 PTGS1 (0.54) RXFP1PTGS1PTGS2KDM4ETDP1
SCHEMBL30556624 0.70 PTGS1 (0.54) RXFP1PTGS1PTGS2KDM4ETDP1
SCHEMBL8373781 0.70 PTGS1 (0.54) RXFP1PTGS1PTGS2KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0370381-B1 2(1H)-quinolinone compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-05-10 EP disclosed
US-4988698-A Cardiovascular disorders, hypotensive agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-01-29 US disclosed
EP-0370381-A2 2(1H)-quinolinone compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-05-30 EP disclosed