SCHEMBL7269198

SCHEMBL7269198

CC(C)(C)OC(=O)NC1CCC(O)C[C@@H]1NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.46
KDM1A O60341 2/20 0.43
GAA P10253 2/20 0.42
MAOB P27338 2/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
CTSK P43235 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
EPHX1 P07099 1/20 0.38
MAOA P21397 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CYP2C9 P11712 1/20 0.36
HSD11B1 P28845 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12096427 1.00 BTK (0.46) BTKKDM1AGAAMAOBNFKB1
SCHEMBL4083324 1.00 BTK (0.46) BTKKDM1AGAAMAOBNFKB1
SCHEMBL3305502 1.00 BTK (0.46) BTKKDM1AGAAMAOBNFKB1
SCHEMBL765258 1.00 BTK (0.46) BTKKDM1AGAAMAOBNFKB1
SCHEMBL13378898 1.00 BTK (0.46) BTKKDM1AGAAMAOBNFKB1
SCHEMBL4367463 0.94 BTK (0.46) BTKKDM1AGAAMAOBNFKB1
SCHEMBL4367460 0.94 BTK (0.46) BTKKDM1AGAAMAOBNFKB1
SCHEMBL17961679 0.94 BTK (0.46) BTKKDM1AGAAMAOBNFKB1
SCHEMBL1988095 0.89 BTK (0.47) BTKKDM1AGAAMAOBNFKB1
SCHEMBL4713065 0.88 BTK (0.45) BTKKDM1AGAAMAOBNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270557-B1 ETHYLENEDIAMINE DERIVATIVES DAIICHI SANKYO CO LTD (JP) 2012-07-25 EP disclosed
EP-1270557-A1 ETHYLENEDIAMINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-01-02 EP disclosed