SCHEMBL7271065

SCHEMBL7271065

COc1ccc(-c2nc3cnccc3[nH]2)c(OCC[S+](C)[O-])c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.44
PDE5A O76074 6/20 0.42
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
AURKA O14965 2/20 0.39
KDR P35968 2/20 0.39
AMY1A P0DUB6 4/20 0.38
ACHE P22303 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
RUNX1 Q01196 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10416712 0.95 PDE2A (0.43) PDE2APDE5APDE3BPDE3ACYP11B1
SCHEMBL7271969 0.92 PDE5A (0.45) PDE2APDE5APDE3BPDE3AAURKA
SCHEMBL10961738 0.91 AURKA (0.39) PDE2APDE5APDE3BPDE3ACYP11B1
SCHEMBL7281143 0.90 PDE2A (0.43) PDE2APDE5APDE3BPDE3ACYP11B1
SCHEMBL7278114 0.88 PDE5A (0.42) PDE5APDE3BPDE3AACHENPC1
SCHEMBL7272240 0.88 PDE2A (0.43) PDE2APDE5APDE3BPDE3ACYP11B1
SCHEMBL10416978 0.87 PDE5A (0.43) PDE2APDE5APDE3BPDE3ACYP11B1
SCHEMBL10416976 0.87 PDE5A (0.45) PDE2APDE5APDE3BPDE3AAURKA
SCHEMBL7271814 0.87 PDE5A (0.41) PDE5APDE3BPDE3AKDRAMY1A
SCHEMBL7282250 0.87 PDE5A (0.41) PDE5APDE3BPDE3AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4904785-A INOTROPIC AGENTS FOR CARDIOVASCULAR DISORDERS ELI LILLY AND COMPANY (US) 1990-02-27 US disclosed
US-4758574-A 2-phenylimidazio (4,5-c) pyridines ELI LILLY AND COMPANY (US) 1988-07-19 US disclosed
EP-0093593-A2 Pyridine compounds ELI LILLY AND COMPANY (US) 1983-11-09 EP disclosed