SCHEMBL7271815

SCHEMBL7271815

CCc1noc(C2=C(C)NC(C)=C(OC(=O)OCCOC)C2c2ccc(Cl)cc2Cl)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.36
PTGDR Q13258 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
RECQL P46063 1/20 0.35
CYP2C9 P11712 3/20 0.34
MEN1 O00255 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 2/20 0.34
KMT2A Q03164 2/20 0.34
HIF1A Q16665 2/20 0.34
HSD17B10 Q99714 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 1/20 0.34
TP53 P04637 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7265677 0.89 CYP2C9 (0.46) KDM4EALDH1A1CYP2C9MEN1CYP1A2
SCHEMBL10995927 0.89 KDM4E (0.46) MAPK1PTGDRPTGDR2KDM4EALDH1A1
SCHEMBL7265650 0.86 ABCC1 (0.32) MAPK1KDM4EALDH1A1RECQLCYP2C9
SCHEMBL7270521 0.86 KMT2A (0.35) MAPK1KDM4EALDH1A1RECQLCYP2C9
SCHEMBL7264418 0.85 KDM4E (0.33) KDM4EALDH1A1MEN1KMT2AHSD17B10
SCHEMBL7263910 0.82 POLB (0.41) MAPK1ALDH1A1CYP2C9MEN1CYP1A2
SCHEMBL7265647 0.81 KMT2A (0.35) MAPK1KDM4EALDH1A1CYP2C9MEN1
SCHEMBL7271627 0.80 CYP2C9 (0.47) KDM4EALDH1A1CYP2C9MEN1CYP1A2
SCHEMBL7265522 0.80 CYP2C9 (0.42) MAPK1KDM4EALDH1A1CYP2C9MEN1
SCHEMBL7271866 0.80 CYP2C9 (0.46) KDM4EALDH1A1CYP2C9MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116708-A1 Substituted 1,4-dihydropyridines, method for their preparation and their use as pharmaceuticals CASSELLA Aktiengesellschaft (DE) 1984-08-29 EP disclosed