SCHEMBL7274263

SCHEMBL7274263

COc1ccc(CC#N)c(Cc2ccccc2)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HTT P42858 2/20 0.44
GAA P10253 1/20 0.44
HTR1A P08908 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7279399 0.87 SLC2A1 (0.49) POLBSMN1; SMN2ABCB1ABCG2HPGD
SCHEMBL10648349 0.83 AOC3 (0.39) POLBSMN1; SMN2KDM4EALDH1A1SLC2A1
SCHEMBL7274621 0.81 POLB (0.52) POLBSMN1; SMN2KDM4EALDH1A1HTT
SCHEMBL7273837 0.80 SLC2A1 (0.42) POLBSMN1; SMN2KDM4EALDH1A1SLC2A1
SCHEMBL28771054 0.79 AOC3 (0.36) POLBSMN1; SMN2KDM4EALDH1A1SLC2A1
SCHEMBL8248932 0.79 BCHE (0.48) POLBSMN1; SMN2KDM4EHTR1AADRA1D
SCHEMBL7281431 0.78 TAAR1 (0.50)
SCHEMBL7283185 0.78 AOC3 (0.39) POLBSMN1; SMN2KDM4EALDH1A1SLC2A1
Hydrochloric Acid SCHEMBL10536541 0.77 TAAR1 (0.49)
SCHEMBL7286452 0.77 SLC2A1 (0.45) POLBSMN1; SMN2KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4885313-A 3,4-Dihydroxyphenylethylamine derivatives and their use FISONS PLC (GB) 1989-12-05 US disclosed
US-4803225-A Dihydroxy-phenethylamino compounds useful as pharmaceuticals FISONS, PLC (GB) 1989-02-07 US disclosed
US-4720586-A Substituted 3,4-dihydroxy-phenylethylamino compounds FISONS, PLC (GB) 1988-01-19 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed