SCHEMBL7274993

SCHEMBL7274993

CC(C)(C)OC(=O)NC(Cc1ccccc1)C(O)C1CCCN1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.55
BACE1 P56817 2/20 0.54
ATM Q13315 1/20 0.47
CTSL P07711 2/20 0.46
REN P00797 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
CTSS P25774 2/20 0.45
CTSB P07858 1/20 0.45
CTSK P43235 1/20 0.45
ACE P12821 2/20 0.45
APP P05067 1/20 0.44
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44
PSENEN Q9NZ42 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8281497 0.94 KLK5 (0.51) KLK5BACE1ATMCTSLREN
SCHEMBL3036976 0.94 KLK5 (0.51) KLK5BACE1ATMCTSLREN
SCHEMBL13390560 0.94 KLK5 (0.51) KLK5BACE1ATMCTSLREN
SCHEMBL7356966 0.83 KLK5 (0.59) KLK5ATMCTSLRENL3MBTL1
Hydrochloric Acid SCHEMBL4365127 0.82 BACE1 (0.58) BACE1
Hydrochloric Acid SCHEMBL4365118 0.82 BACE1 (0.58) BACE1
Hydrochloric Acid SCHEMBL4365123 0.82 BACE1 (0.58) BACE1
SCHEMBL6446193 0.80 KLK5 (0.63) KLK5ATMCTSLCTSSCTSB
SCHEMBL6445261 0.80 KLK5 (0.63) KLK5ATMCTSLCTSSCTSB
SCHEMBL6444857 0.80 KLK5 (0.63) KLK5ATMCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0361341-A2 Therapeutics for aids based on inhibitors of HIV protease MILES INC. (US) 1990-04-04 EP disclosed