SCHEMBL7275334

SCHEMBL7275334

COCCOC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1cccc(Cl)c1Cl

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.70
MEN1 O00255 3/20 0.70
CYP1A2 P05177 3/20 0.70
CYP3A4 P08684 3/20 0.70
CYP2C19 P33261 3/20 0.70
KMT2A Q03164 3/20 0.70
ABCB11 O95342 3/20 0.70
TBXA2R P21731 3/20 0.70
ADRA1A P35348 3/20 0.70
SLC6A3 Q01959 3/20 0.70
TSHR P16473 3/20 0.70
KDM4E B2RXH2 2/20 0.70
HIF1A Q16665 2/20 0.70
HSD17B10 Q99714 2/20 0.70
ABCB1 P08183 2/20 0.70
ADORA3 P0DMS8 2/20 0.70
ADRB3 P13945 2/20 0.70
OPRK1 P41145 2/20 0.70
SCN5A Q14524 2/20 0.70
CYP2D6 P10635 2/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7407254 0.92 CYP2C9 (0.83) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL10410007 0.91 CYP2C9 (0.67) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL7074057 0.91 CYP2C9 (0.70) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL7267278 0.91 CYP2C9 (0.57) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL7265394 0.90 CYP2C9 (0.82) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL8084216 0.88 CYP2C9 (0.64) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL7421000 0.88 CYP2C9 (0.63) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL7410229 0.88 CYP2C9 (0.66) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL7407221 0.88 CYP2C9 (0.66) CYP2C9MEN1CYP1A2CYP3A4CYP2C19
SCHEMBL820019 0.87 KDM4E (0.78) CYP2C9MEN1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4920225-A Resolution of 1,4-dihydropyridine derivatives LABORATOIRES SYNTEX S.A. (FR) 1990-04-24 US disclosed
EP-0273349-A2 Resolution of 1,4-dihydropyridine derivatives LABORATOIRES SYNTEX S.A. (FR) 1988-07-06 EP disclosed