SCHEMBL7276002

SCHEMBL7276002

CC(C)(C)OC(=O)NC(Cc1cscn1)C(O)C(O)C(Cc1cscn1)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.44
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CTSK P43235 4/20 0.38
CTSS P25774 2/20 0.38
PTPRB P23467 4/20 0.37
KLK5 Q9Y337 2/20 0.37
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
ATM Q13315 1/20 0.35
CA4 P22748 1/20 0.35
CA9 Q16790 1/20 0.35
CYP2D6 P10635 1/20 0.35
TRPA1 O75762 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339982 1.00 SCN9A (0.44) SCN9ACA1CA2CA7CTSK
SCHEMBL6730949 0.84 SCN9A (0.46) SCN9ACA1CA2CA7CTSK
SCHEMBL6747611 0.82 SCN9A (0.44) SCN9ACA1CA2CA7CTSK
SCHEMBL478732 0.82 SCN9A (0.53) SCN9ACTSKCTSSITGB3ITGA2B
SCHEMBL8245755 0.82 SCN9A (0.44) SCN9ACA1CA2CA7CTSK
SCHEMBL478735 0.82 SCN9A (0.53) SCN9ACTSKCTSSITGB3ITGA2B
SCHEMBL5717580 0.82 SCN9A (0.53) SCN9ACTSKCTSSITGB3ITGA2B
SCHEMBL23324594 0.81 SCN9A (0.50) SCN9ACTSKCTSSPTPRBKLK5
Hydrochloric Acid SCHEMBL28584085 0.81 SCN9A (0.52) SCN9ACTSKCTSSITGB3ITGA2B
SCHEMBL9439647 0.81 SCN9A (0.44) SCN9ACA1CA2CA7CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed