SCHEMBL728142

SCHEMBL728142

CC1=CCC(c2nn(C(C)(C)CN/C(=N/C(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)c3ncnc(N)c23)C=C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 6/20 0.57
RIPK2 O43353 2/20 0.40
SRC P12931 6/20 0.34
PTK6 Q13882 6/20 0.34
HCK P08631 3/20 0.34
FYN P06241 2/20 0.34
BLK P51451 2/20 0.34
LCK P06239 1/20 0.34
LYN P07948 1/20 0.34
FRK P42685 1/20 0.34
ABL1 P00519 9/20 0.33
KDR P35968 4/20 0.33
EGFR P00533 4/20 0.33
PIK3CD O00329 3/20 0.33
PIK3CA P42336 3/20 0.33
PIK3CG P48736 3/20 0.33
PRKDC P78527 3/20 0.33
PI4KB Q9UBF8 2/20 0.33
BACE1 P56817 1/20 0.33
PIK3CB P42338 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL726560 0.84 RET (0.69) RETRIPK2SRCPTK6FYN
SCHEMBL728046 0.81 RET (0.69) RETRIPK2SRCPTK6FYN
SCHEMBL727071 0.81 RET (0.53) RETRIPK2KDREGFRBTK
SCHEMBL727933 0.80 RET (0.62) RETRIPK2SRCABL1KDR
SCHEMBL726637 0.80 RET (0.76) RETRIPK2SRCPTK6HCK
SCHEMBL728198 0.79 RIPK2 (0.64) RETRIPK2SRCPTK6HCK
SCHEMBL19265932 0.79 RIPK2 (0.64) RETRIPK2SRCPTK6HCK
SCHEMBL10098363 0.79 RET (0.61) RETRIPK2SRCABL1KDR
SCHEMBL726543 0.78 RET (0.80) RETRIPK2SRCPTK6HCK
SCHEMBL726555 0.78 RET (0.60) RETRIPK2SRCABL1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003544-A1 PROTEIN KINASE INHIBITORS AND METHODS OF TREATMENT THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2012-01-12 WO disclosed