SCHEMBL7282005

SCHEMBL7282005

CCCCCNN(C)NCCCCC

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
ALDH1A1 P00352 1/20 0.50
EPHX1 P07099 7/20 0.46
ADH1B P00325 2/20 0.40
ADH1C P00326 2/20 0.40
ADH1A P07327 2/20 0.40
ADH7 P40394 2/20 0.40
ADH4 P08319 1/20 0.40
DNM1 Q05193 3/20 0.39
THRB P10828 1/20 0.39
PPARA Q07869 2/20 0.36
GBA1 P04062 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29658268 0.97 EPHX1 (0.50) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL30368694 0.91 TSHR (0.43) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL578890 0.82
SCHEMBL258474 0.80 EPHX1 (0.50) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL578496 0.80 EPHX1 (0.50) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL258725 0.80 EPHX1 (0.50) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL11862257 0.80 EPHX1 (0.50) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL1903292 0.80 EPHX1 (0.50) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL258373 0.80 EPHX1 (0.50) TSHRALDH1A1EPHX1ADH1BADH1C
SCHEMBL464960 0.80 EPHX1 (0.50) TSHRALDH1A1EPHX1ADH1BADH1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422937-B1 Fibrinogen receptor antagonists MERCK & CO INC (US) 1994-03-02 EP claimed
EP-0422938-B1 Fibrinogen receptor antagonists MERCK & CO INC (US) 1995-02-22 EP disclosed
US-5374622-A Modified cyclic heptapeptides MERCK & CO., INC. (US) 1994-12-20 US disclosed
US-5338723-A Anticoagulants and thrombus preventatives comprising cyclic hexapeptides having a synthetic amino acid replace arginine in the sequence of arginine/glycine/aspartic acid MERCK & CO., INC. (US) 1994-08-16 US disclosed
EP-0422937-B1 Fibrinogen receptor antagonists MERCK & CO INC (US) 1994-03-02 EP disclosed
EP-0422938-A1 Fibrinogen receptor antagonists MERCK & CO. INC. (US) 1991-04-17 EP disclosed
EP-0422937-A1 Fibrinogen receptor antagonists MERCK & CO. INC. (US) 1991-04-17 EP disclosed