SCHEMBL7284686

SCHEMBL7284686

COC(=O)C[C@H](N)CCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.49
S1PR2 O95136 1/20 0.49
S1PR1 P21453 1/20 0.49
METAP2 P50579 1/20 0.48
METAP1 P53582 1/20 0.48
TSHR P16473 1/20 0.47
CTSG P08311 1/20 0.47
CTRB1 P17538 1/20 0.47
ANPEP P15144 2/20 0.46
ERAP1 Q9NZ08 2/20 0.46
ERAP2 Q6P179 1/20 0.46
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
MMP12 P39900 1/20 0.46
MEN1 O00255 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8170979 1.00 DPP4 (0.49) DPP4S1PR2S1PR1METAP2METAP1
SCHEMBL8170975 1.00 DPP4 (0.49) DPP4S1PR2S1PR1METAP2METAP1
Hydrochloric Acid SCHEMBL7284681 0.98 DPP4 (0.48) DPP4S1PR2S1PR1METAP2METAP1
Hydrochloric Acid SCHEMBL7274932 0.98 DPP4 (0.48) DPP4S1PR2S1PR1METAP2METAP1
Acetic Acid SCHEMBL7371940 0.97 DPP4 (0.47) DPP4S1PR2S1PR1METAP2METAP1
Acetic Acid SCHEMBL7374879 0.97 DPP4 (0.47) DPP4S1PR2S1PR1METAP2METAP1
Acetic Acid SCHEMBL7371937 0.97 DPP4 (0.47) DPP4S1PR2S1PR1METAP2METAP1
SCHEMBL2311407 0.84 F2 (0.55) DPP4S1PR2S1PR1TSHRMEN1
SCHEMBL8903673 0.84 F2 (0.55) DPP4S1PR2S1PR1TSHRMEN1
SCHEMBL6343323 0.83 EPHX1 (0.53) DPP4ANPEPSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114328-A ANTICOAGULANTS; BLOOD DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-09-05 US disclosed
EP-0512831-B1 Fibrinogen receptor antagonists MERCK & CO INC (US) 1999-09-22 EP disclosed
US-5849736-A Isoxazoline and isoxazole fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-12-15 US disclosed
US-5455243-A Anticoagulants MERCK & CO., INC. (US) 1995-10-03 US disclosed
US-5281585-A Secondary amide containing antagonist MERCK & CO., INC. (US) 1994-01-25 US disclosed
WO-1992019595-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1992-11-12 WO disclosed
EP-0512831-A1 Fibrinogen receptor antagonists MERCK & CO. INC. (US) 1992-11-11 EP disclosed
US-4585887-A Process for the production of optically active 3-aminocarboxylic acid esters LONZA LTD. (CH) 1986-04-29 US disclosed