SCHEMBL7286552

SCHEMBL7286552

CCOCN1C(C)=C(C(=O)O)C(c2cccc([N+](=O)[O-])c2)C(C(=O)O)=C1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.57
CYP3A4 P08684 3/20 0.57
CYP2C9 P11712 3/20 0.57
CYP2C19 P33261 3/20 0.57
MAPT P10636 3/20 0.57
CYP2D6 P10635 2/20 0.57
TSHR P16473 2/20 0.57
NFKB1 P19838 2/20 0.57
LMNA P02545 2/20 0.57
GMNN O75496 1/20 0.57
BLM P54132 1/20 0.57
PMP22 Q01453 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
CACNA1F O60840 10/20 0.56
CACNA1D Q01668 10/20 0.56
CACNA1S Q13698 10/20 0.56
CACNA1C Q13936 10/20 0.56
ADORA3 P0DMS8 1/20 0.56
HIF1A Q16665 3/20 0.53
MEN1 O00255 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7286542 1.00 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9123056 0.95 CYP1A2 (0.66) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9032405 0.94 CYP1A2 (0.67) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL10391376 0.94 CYP1A2 (0.67) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL7275483 0.94 CYP1A2 (0.67) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL11688660 0.92 CYP1A2 (0.55) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL11688678 0.92 CYP1A2 (0.55) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL11687260 0.90 MAPT (0.70) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL11687126 0.89 CYP1A2 (0.56) CYP1A2CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL9033028 0.89 CYP1A2 (0.72) CYP1A2CYP3A4CYP2C9CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0494816-B1 1,4-Dihydropyridine derivatives, process for their preparation and therapeutical composition containing them LAFON LABOR (FR) 1999-07-21 EP disclosed
US-5475111-A Process for the preparation of dihydropyridinecarboxylic acids BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1995-12-12 US disclosed
US-4994461-A Vasodilators; treating cardiovascular disorders BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1991-02-19 US disclosed
EP-0240398-A1 Dissymmetrical 1,4-dihydropyridine-3,5-dicarboxylic-acid derivatives, preparation processes and therapeutical use FOURNIER INNOVATION ET SYNERGIE (FR) 1987-10-07 EP disclosed
US-4021434-A CEREBRAL VASODILATORS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JA) 1977-05-03 US disclosed