SCHEMBL7287552

SCHEMBL7287552

Nc1ccc(C2=NNC(=O)CO2)cc1

nearest known ligand 0.61

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
MAOB P27338 20/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22288623 0.84 MAOB (0.63) MAOB
SCHEMBL22304501 0.83 MAOB (0.63) MAOB
SCHEMBL517561 0.82 MAOB (0.74) MAOB
SCHEMBL9667797 0.82 MAOB (0.57) MAOB
SCHEMBL22304755 0.81 MAOB (0.61) MAOB
SCHEMBL10806139 0.81 MAOB (0.56) MAOB
SCHEMBL10800830 0.79 MAOB (0.57) MAOB
SCHEMBL9668897 0.78 MAOB (0.56) MAOB
SCHEMBL22288965 0.76 MAOB (0.56) MAOB
SCHEMBL22304801 0.75 MAOB (0.53) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0383449-B1 Pyridazinone derivatives and processes for preparing the same ORION YHTYMAE OY (FI) 1995-09-06 EP disclosed
US-5185332-A Treating congestive heart failure ORION-YHTYMA OY (FI) 1993-02-09 US disclosed
US-5122524-A Treatment for congestive heart failure; hypertensive agents; vasodilation ORION-YHTYMA OY (FI) 1992-06-16 US disclosed
EP-0223937-B1 INDOLES SUBSTITUTED WITH HETEROCYCLES, INTERMEDIATES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS Roche Diagnostics GmbH (DE) 1992-03-18 EP disclosed
US-5019575-A Congestive Heart Failure Treatment ORION-YHTYMA OY (FI) 1991-05-28 US disclosed
EP-0383449-A2 Pyridazinone derivatives and processes for preparing the same ORION-YHTYMÀ„ OY (FI) 1990-08-22 EP disclosed
US-4851406-A CARDIOVASCULAR DISORDERS, HYPOTENSIVE BOEHRINGER MANNHEIM GMBH (DE) 1989-07-25 US disclosed
US-4683232-A N,N-DIMETHYL-P-(2,3-DIHYDRO-2-OXO-6H-1,3,4 OXADIAZIN-2-YLBENZAMIDE IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-07-28 US disclosed
EP-0223937-A1 Indoles substituted with heterocycles, intermediates, process for their preparation and medicaments Roche Diagnostics GmbH (DE) 1987-06-03 EP disclosed
US-4587246-A CARDIOTONIC IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-05-06 US disclosed
EP-0052442-B1 HETEROCYCLIC COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-09-11 EP disclosed
US-4503054-A VASODILATORS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-03-05 US disclosed
US-4423045-A CARDIOVASCULAR DISORDERS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-12-27 US disclosed
EP-0052442-A1 Heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-05-26 EP disclosed