SCHEMBL7294191

SCHEMBL7294191

COC(=O)[C@@H]1CCCN1C(=O)[C@H]1CCCN1C(=O)CC1CCc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PREP P48147 12/20 0.50
ACE P12821 1/20 0.45
ALDH1A1 P00352 2/20 0.42
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
F2 P00734 1/20 0.41
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294194 1.00 PREP (0.50) PREPACEALDH1A1MAPK1L3MBTL1
SCHEMBL7302938 0.96 PREP (0.48) PREPACEALDH1A1MAPK1L3MBTL1
SCHEMBL7303285 0.87 PREP (0.54) PREPACEALDH1A1F2
SCHEMBL7303289 0.87 PREP (0.54) PREPACEALDH1A1F2
SCHEMBL7298496 0.84 PREP (0.71) PREPF2
SCHEMBL7298505 0.84 PREP (0.71) PREPF2
SCHEMBL7300348 0.84 PREP (0.53) PREPF2
SCHEMBL7301748 0.84 PREP (0.70) PREP
SCHEMBL7301742 0.84 PREP (0.70) PREP
SCHEMBL7296462 0.83 PREP (0.52) PREPF2PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017929-A Cholinesterase activator ZERIA PHARMACEUTICAL CO., LTD. (JP) 2000-01-25 US disclosed
EP-0754454-A1 CHOLINESTERASE ACTIVATOR ZERIA PHARMACEUTICAL CO., LTD. (JP) 1997-01-22 EP disclosed
EP-0372484-B1 Condensed benzene derivative ZERIA PHARM CO LTD (JP) 1994-10-26 EP disclosed
US-5028604-A Cognition Activators ZERIA PHARMACEUTICAL CO., LTD. (JP) 1991-07-02 US disclosed
EP-0372484-A2 Condensed benzene derivative ZERIA PHARMACEUTICAL CO., LTD. (JP) 1990-06-13 EP disclosed