SCHEMBL7296380

SCHEMBL7296380

C=COC(=O)N1C2CCC1CC(OC(=O)c1cc(Cl)cc(Cl)c1)C2

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.63
HTR3E A5X5Y0 3/20 0.63
HTR3B O95264 3/20 0.63
HTR3A P46098 3/20 0.63
HTR3D Q70Z44 3/20 0.63
HTR3C Q8WXA8 3/20 0.63
CYP1A2 P05177 2/20 0.63
GMNN O75496 1/20 0.63
ALOX15 P16050 1/20 0.63
TSHR P16473 1/20 0.63
MTOR P42345 1/20 0.63
PMP22 Q01453 1/20 0.63
HSD17B10 Q99714 1/20 0.63
GAA P10253 1/20 0.62
CYP2C19 P33261 2/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
NR1I2 O75469 1/20 0.45
POLB P06746 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7304481 0.79 CYP2D6 (0.67) CYP2D6HTR3EHTR3BHTR3AHTR3D
Bemesetron SCHEMBL195147 0.78 CYP2D6 (1.00) CYP2D6HTR3EHTR3BHTR3AHTR3D
Bemesetron SCHEMBL29430183 0.78 CYP2D6 (1.00) CYP2D6HTR3EHTR3BHTR3AHTR3D
Bemesetron SCHEMBL195148 0.78 CYP2D6 (1.00) CYP2D6HTR3EHTR3BHTR3AHTR3D
Bemesetron SCHEMBL10765684 0.78 CYP2D6 (1.00) CYP2D6HTR3EHTR3BHTR3AHTR3D
Bemesetron SCHEMBL5790539 0.78 CYP2D6 (1.00) CYP2D6HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL7299830 0.78 GAA (0.72) CYP2D6HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL7293406 0.78 GAA (0.68) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL7291276 0.77 CYP2D6 (0.69) CYP2D6HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL7295017 0.76 GAA (0.70) CYP2D6HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5252570-A Amidino and guanidino derivatives B.I. ITALIA (IT) 1993-10-12 US disclosed
US-5047410-A Indolyl derivatives and their use as 5-HT3, receptor antagonists ISTITUTO DE ANGELI S.P.A. (IT) 1991-09-10 US disclosed
EP-0351385-A2 New amidino and guanidino derivatives BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1990-01-17 EP disclosed