SCHEMBL7300349

SCHEMBL7300349

Cc1ccc2c(c1)OC(C)(C)C[CH]2

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.33
HTR1A P08908 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
TRPA1 O75762 2/20 0.32
CNR1 P21554 2/20 0.32
CNR2 P34972 2/20 0.32
TRPV1 Q8NER1 2/20 0.32
TRPV3 Q8NET8 2/20 0.32
TRPV4 Q9HBA0 2/20 0.32
TRPV2 Q9Y5S1 2/20 0.32
KDM4E B2RXH2 3/20 0.31
HTT P42858 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MMP12 P39900 1/20 0.31
MAOB P27338 1/20 0.31
CA12 O43570 1/20 0.31
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7293466 0.85 KDM4E (0.34) SLC6A2HTR1AHTR2CHTR2BSIGMAR1
SCHEMBL7298544 0.80 HTR2C (0.44) HTR2CMAOBCA12CA9
SCHEMBL7293318 0.80 HTR2C (0.42) HTR2CKDM4EHTTALDH1A1LMNA
SCHEMBL7290026 0.80 HTR2C (0.42) HTR2CMAOB
SCHEMBL9583438 0.77 HTR2C (0.47) HTR1AHTR2CHTR2BSIGMAR1TRPA1
SCHEMBL9583946 0.76 DAO (0.33) TRPV1LMNACA9TP53
SCHEMBL7300321 0.76 ABCB1 (0.38) KDM4ELMNAMAOBCA12CA9
SCHEMBL7299822 0.75 AKR1B1 (0.43) ALDH1A1LMNACA12CA9CYP3A4
SCHEMBL1707125 0.75 MEN1 (0.40) HTR2CHTR2BTP53
SCHEMBL3535518 0.74 CYP3A4 (0.33) KDM4EHTTALDH1A1MAOBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260444-A Cardiovascular, hypotensive WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed
US-5208245-A Hypotensive agents WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-05-04 US disclosed
EP-0460418-A2 Novel Dihydropyridine derivative WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1991-12-11 EP disclosed