SCHEMBL7300690

SCHEMBL7300690

COc1ccc(C2CNC(=O)C2)cc1Br

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 18/20 0.76
PDE4B Q07343 12/20 0.76
PDE4C Q08493 12/20 0.76
PDE4D Q08499 12/20 0.76
CYP3A4 P08684 2/20 0.63
ALDH1A1 P00352 2/20 0.63
CYP1A2 P05177 2/20 0.63
VEGFA P15692 1/20 0.63
LMNA P02545 1/20 0.63
MAPT P10636 1/20 0.63
CYP2C9 P11712 1/20 0.63
ALOX15 P16050 1/20 0.63
CREBBP Q92793 1/20 0.63
KDM4E B2RXH2 1/20 0.63
PDE5A O76074 1/20 0.63
TNF P01375 1/20 0.63
MAPK1 P28482 1/20 0.63
BLM P54132 1/20 0.63
PDE1A P54750 1/20 0.63
PDE1B Q01064 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7293719 0.87 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL22562810 0.84 PDE4A (0.78) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL13677704 0.83 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL22562815 0.83 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL9792208 0.83 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL3541828 0.83 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL18117803 0.83 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL9647066 0.83 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL19559499 0.83 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL23118946 0.81 PDE4A (0.72) PDE4APDE4BPDE4CPDE4DCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0350437-B1 3,4-Disubstituted phenyl-heterocycles and their use SCHERING AG (DE) 1995-09-06 EP disclosed
US-5064854-A 3,4-DISUBSTITUTED PHENYL HETEROCYCLES AND THEIR USE SCHERING AKTIENGESELLSCHAFT (DE) 1991-11-12 US disclosed
EP-0350437-A1 3,4-Disubstituted phenyl-heterocycles and their use SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-10 EP disclosed