SCHEMBL7301302

SCHEMBL7301302

CCc1nc(-c2ccc(OCCCN3CCN(C)CC3)cc2)no1

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 8/20 0.69
ACACB O00763 2/20 0.64
ACACA Q13085 2/20 0.64
RAB9A P51151 2/20 0.55
NPC1 O15118 1/20 0.55
DRD3 P35462 2/20 0.50
KDM4E B2RXH2 1/20 0.50
HRH3 Q9Y5N1 4/20 0.49
MAPK1 P28482 1/20 0.49
USP2 O75604 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
HRH4 Q9H3N8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7293044 0.91 ACACB (0.64) CXCR1ACACBACACARAB9ANPC1
SCHEMBL7327061 0.90 ACACB (0.62) CXCR1ACACBACACARAB9ANPC1
SCHEMBL7295131 0.80 ACACB (0.97) ACACBACACARAB9ANPC1MAPK1
SCHEMBL7292052 0.78 ACACB (0.62) CXCR1ACACBACACARAB9ANPC1
SCHEMBL17233279 0.78 ACACB (0.73) ACACBACACARAB9ANPC1MAPK1
SCHEMBL3503745 0.77 ACACB (0.61) ACACBACACAKDM4EHRH3ALDH1A1
SCHEMBL18598419 0.77 ACACB (0.71) ACACBACACARAB9ANPC1MAPK1
SCHEMBL7291741 0.76 HPGD (0.64) ACACBACACARAB9AKDM4EMAPK1
SCHEMBL23588222 0.76 ACACB (0.70) CXCR1ACACBACACARAB9ANPC1
SCHEMBL7302028 0.76 ACACB (0.70) ACACBACACARAB9ANPC1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0504574-B1 1,2,4-Oxadiazole derivatives having monoamine oxidase B enzyme-inhibitory activity and method for preparing same WAKAMOTO PHARMA CO LTD (JP) 1996-02-28 EP disclosed
US-5356916-A Treating Parkinson*s disease WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1994-10-18 US disclosed
EP-0504574-A1 1,2,4-Oxadiazole derivatives having monoamine oxidase B enzyme-inhibitory activity and method for preparing same Wakamoto Pharmaceutical Co., Ltd. (JP) 1992-09-23 EP disclosed