SCHEMBL7301581

SCHEMBL7301581

O=P(CCc1ccccc1)(OCc1ccccc1)OCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.57
CETP P11597 4/20 0.47
CYP2D6 P10635 1/20 0.43
POLB P06746 1/20 0.42
KLK8 O60259 1/20 0.42
PLAU P00749 1/20 0.42
KLK2 P20151 1/20 0.42
KLK4 Q9Y5K2 1/20 0.42
ACP3 P15309 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14277384 0.89 TSHR (0.50) TSHRCETPCYP2D6KLK8PLAU
SCHEMBL11509944 0.84 CETP (0.49) TSHRCETPCYP2D6KLK8PLAU
SCHEMBL5248630 0.82 CETP (0.47) TSHRCETPPOLB
SCHEMBL5028595 0.82 TSHR (0.60) TSHRCETP
SCHEMBL1243459 0.82 TSHR (0.55) TSHRCETPPOLB
SCHEMBL5404588 0.82 CETP (0.58) TSHRCETP
SCHEMBL5327008 0.81 TSHR (0.63) TSHRCETP
SCHEMBL13896611 0.81 TSHR (0.53) TSHRCETPCYP2D6POLB
SCHEMBL4154482 0.81 TSHR (0.53) TSHRCETPPOLB
SCHEMBL11148077 0.79 TSHR (0.52) TSHRCETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4963539-A TREATING HEART FAILURE, PAIN OR DIARRHEA E. R. SQUIBB & SONS, INC. (US) 1990-10-16 US disclosed
EP-0306879-A2 Phosphonate and phosphonamide endopeptidase inhibitors E.R. SQUIBB & SONS, INC. (US) 1989-03-15 EP disclosed