SCHEMBL7301768

SCHEMBL7301768

CCn1c(=O)c2[nH]c(C=Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)nc2n(CC)c1=O

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.49
SIRT2 Q8IXJ6 1/20 0.46
SIRT1 Q96EB6 1/20 0.46
SIRT3 Q9NTG7 1/20 0.46
SIRT5 Q9NXA8 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301754 1.00 ADORA2A (0.49) ADORA2ASIRT2SIRT1SIRT3SIRT5
SCHEMBL7315930 0.89 ADORA2A (0.63) ADORA2AADORA2BADORA1
SCHEMBL7315934 0.89 ADORA2A (0.63) ADORA2AADORA2BADORA1
SCHEMBL7306207 0.89 KDM4E (0.47) ADORA2ASIRT2SIRT1SIRT3SIRT5
SCHEMBL7306221 0.89 KDM4E (0.47) ADORA2ASIRT2SIRT1SIRT3SIRT5
SCHEMBL7309799 0.85 SIRT2 (0.49) SIRT2SIRT1SIRT3SIRT5ADORA2B
SCHEMBL7309789 0.85 SIRT2 (0.49) SIRT2SIRT1SIRT3SIRT5ADORA2B
SCHEMBL7309857 0.81
SCHEMBL7309870 0.81
SCHEMBL7315254 0.81 ADORA2A (0.48) ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628311-B1 Xanthine-Derivatives as Antidepressants KYOWA HAKKO KOGYO KK (JP) 2002-04-24 EP disclosed
US-5587378-A ADMINISTERING A SUBSTITUTED XANTHINE COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-12-24 US disclosed
US-5543415-A ADMINISTERING A XANTHINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-08-06 US disclosed
US-5484920-A XANTHINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-01-16 US disclosed
EP-0628311-A1 ANTIDEPRESSANT KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-12-14 EP disclosed
EP-0590919-A1 Therapeutic agents for parkinson's disease KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-04-06 EP disclosed