SCHEMBL7303267

SCHEMBL7303267

Cc1ccc(S(=O)(=O)O[C@@H]2C[C@@H](C(=O)NC(C)(C)C)N(C(=O)OC(C)(C)C)C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 13/20 0.47
CYP1A2 P05177 1/20 0.46
POLB P06746 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSD11B1 P28845 1/20 0.44
BCL2 P10415 2/20 0.42
BCL2L1 Q07817 2/20 0.42
F13A1 P00488 1/20 0.41
TGM2 P21980 1/20 0.41
TGM1 P22735 1/20 0.41
LMNA P02545 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3182745 0.88 NR1H2 (0.47) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL6847610 0.88 NR1H2 (0.47) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL8166919 0.88 NR1H2 (0.47) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL6847613 0.88 NR1H2 (0.47) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL2819569 0.88 NR1H2 (0.47) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL25097911 0.88 NR1H2 (0.47) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL6847935 0.88 NR1H2 (0.47) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL4320166 0.88 NR1H2 (0.47) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL6847660 0.87 MCL1 (0.46) MCL1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL13481726 0.87 MCL1 (0.44) MCL1CYP1A2POLBCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed