SCHEMBL7303683

SCHEMBL7303683

Cc1cnc(COC(=O)NC(C(=O)O)C(C)C)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 3/20 0.46
NPSR1 Q6W5P4 1/20 0.39
ECE1 P42892 2/20 0.38
MME P08473 1/20 0.38
CASP1 P29466 1/20 0.38
CASP3 P42574 1/20 0.38
CASP7 P55210 1/20 0.38
CASP6 P55212 1/20 0.38
CASP8 Q14790 1/20 0.38
CTSL P07711 2/20 0.37
CTSB P07858 2/20 0.37
CTSK P43235 2/20 0.37
CTSS P25774 1/20 0.37
GPR132 Q9UNW8 2/20 0.36
POLB P06746 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
MBTPS1 Q14703 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303687 1.00 TYR (0.46) TYRNPSR1ECE1MMECASP1
SCHEMBL7304330 0.82 TYR (0.46) TYRNPSR1ECE1MMECTSL
SCHEMBL7304329 0.82 TYR (0.46) TYRNPSR1ECE1MMECTSL
SCHEMBL7303476 0.81 TYR (0.46) TYRNPSR1ECE1MMECASP1
SCHEMBL7303468 0.81 TYR (0.46) TYRNPSR1ECE1MMECASP1
SCHEMBL7303071 0.78 TYR (0.46) TYRECE1MMECTSLCTSB
SCHEMBL7298552 0.78 TYR (0.46) TYRECE1MMECTSLCTSB
SCHEMBL3033874 0.76 NPC1 (0.59) TYRECE1MMECTSLCTSB
SCHEMBL4675990 0.76 NPC1 (0.59) TYRECE1MMECTSLCTSB
SCHEMBL7395887 0.75 TYR (0.48) TYRNPSR1ECE1MMECTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed