SCHEMBL7304399

SCHEMBL7304399

Cn1cnc2ncnc-2c1Cl

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
YTHDC1 Q96MU7 1/20 0.32
CDK1 P06493 1/20 0.31
DYRK1A Q13627 1/20 0.30
KDM5A P29375 1/20 0.30
KDM4C Q9H3R0 1/20 0.30
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1914 0.75 ADORA2A (0.41) ADORA2AADORA1YTHDC1CDK1DYRK1A
SCHEMBL1997511 0.72 ADORA2A (0.32) ADORA2AADORA1YTHDC1
SCHEMBL360582 0.67
SCHEMBL19059638 0.64
SCHEMBL5387153 0.64
SCHEMBL15842953 0.63
SCHEMBL21719978 0.61 KDM4E (0.42) KDM4EYTHDC1CDK1
SCHEMBL14732773 0.61 KDM4E (0.42) KDM4EYTHDC1CDK1
SCHEMBL8326360 0.61
SCHEMBL860591 0.60

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5177207-A Cardiac failure, memory defecit HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1993-01-05 US disclosed
US-5145855-A Hypotensive, memory deficit, asthma, psorisis HOECHST ROUSSEL PHARMACEUTICALS, INC. (US) 1992-09-08 US disclosed
US-5093336-A Treatment of cardiac failure and memory deficit HOECHAT-ROUSSEL PHARMACEUTICALS, INC. (US) 1992-03-03 US disclosed
US-4999351-A Treating cardiac failure and memory deficit HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0406789-A1 6-and 7-Deoxyforskolin and derivates thereof, intermediates and a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-09 EP disclosed
EP-0378159-A1 7-Aryl- and heteroaryl ethers of desacetylforskolin, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1990-07-18 EP disclosed