SCHEMBL7304702

SCHEMBL7304702

CCCc1cc(OCC)c2c(c1OC)S(=O)(=O)N(CSc1ccccc1)C2=O

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ELANE P08246 14/20 0.44
HTT P42858 1/20 0.35
EGFR P00533 2/20 0.34
APLNR P35414 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7314724 0.84 ELANE (0.66) ELANE
SCHEMBL7304861 0.81 ELANE (0.37) ELANEHTTMEN1KMT2A
SCHEMBL7309354 0.78 ELANE (0.48) ELANEEGFRAPLNRTSHRKMT2A
SCHEMBL7287449 0.77 ELANE (0.59) ELANE
SCHEMBL7340454 0.76 ELANE (0.49) ELANE
SCHEMBL7286964 0.76 ELANE (0.65) ELANEHTTMEN1KMT2A
SCHEMBL7281488 0.75 ELANE (0.70) ELANEHTTAPLNRMEN1KMT2A
SCHEMBL7282040 0.75 ELANE (0.52) ELANEAPLNRTSHR
SCHEMBL7287974 0.74 ELANE (0.57) ELANETSHR
SCHEMBL7309320 0.74 MAPT (0.44) ELANEHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874432-A Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof SANOFI (FR) 1999-02-23 US disclosed
US-5650422-A TREATMENT OF EMPHYSEMA, ARTHRITIS OR PANCREATITIS SANOFI (FR) 1997-07-22 US disclosed
US-5596012-A Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof STERLING WINTHROP INC. (US) 1997-01-21 US disclosed
US-5371074-A Use of saccharin derivatives as proteolytic enzyme inhibitors STERLING WINTHROP INC. (US) 1994-12-06 US disclosed
US-5236917-A Respiratory system disorders, antiarthritic agents STERLING WINTHROP INC. (US) 1993-08-17 US disclosed
EP-0542372-A1 2-Substituted saccharin derivative proteolytic enzyme inhibitors STERLING WINTHROP INC. (US) 1993-05-19 EP disclosed