SCHEMBL7305744

SCHEMBL7305744

CC(=O)N(C)C1(c2ccccc2)CCN(CCCC2(c3ccc(Cl)c(Cl)c3)CCCNC2)CC1

nearest known ligand 0.72

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 11/20 0.72
TACR2 P21452 10/20 0.72
TACR1 P25103 10/20 0.72
CYP2D6 P10635 2/20 0.72
CYP3A4 P08684 1/20 0.72
CYP2C9 P11712 1/20 0.72
CYP2C19 P33261 1/20 0.72
SLC6A2 P23975 4/20 0.51
SLC6A4 P31645 4/20 0.51
SLC6A3 Q01959 4/20 0.51
CCR5 P51681 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7751688 0.99 TACR3 (0.71) TACR3TACR2TACR1CYP2D6CYP3A4
SCHEMBL17131459 0.86 TACR2 (0.86) TACR3TACR2TACR1CYP2D6CYP3A4
Osanetant SCHEMBL5679271 0.84 TACR2 (1.00) TACR3TACR2TACR1CYP2D6CYP3A4
Osanetant SCHEMBL29371450 0.84 TACR2 (1.00) TACR3TACR2TACR1CYP2D6CYP3A4
Osanetant SCHEMBL119440 0.84 TACR2 (1.00) TACR3TACR2TACR1CYP2D6CYP3A4
Osanetant SCHEMBL30961738 0.84 TACR2 (1.00) TACR3TACR2TACR1CYP2D6CYP3A4
Osanetant SCHEMBL4080131 0.84 TACR2 (1.00) TACR3TACR2TACR1CYP2D6CYP3A4
Osanetant SCHEMBL6543149 0.83 TACR2 (0.98) TACR3TACR2TACR1CYP2D6CYP3A4
Osanetant SCHEMBL5679471 0.83 TACR2 (0.98) TACR3TACR2TACR1CYP2D6CYP3A4
SCHEMBL8136920 0.83 TACR2 (0.95) TACR3TACR2TACR1CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673928-B1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists SANOFI SYNTHELABO (FR) 2001-08-29 EP disclosed
EP-0673928-A1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists SANOFI (FR) 1995-09-27 EP disclosed