SCHEMBL7306608

SCHEMBL7306608

Nc1ccc([O])c(N)c1N

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.36
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
CD44 P16070 1/20 0.32
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
TDP1 Q9NUW8 1/20 0.30
CYP3A4 P08684 1/20 0.30
ALOX15 P16050 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
LMNA P02545 1/20 0.30
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30
BLM P54132 1/20 0.30
HIF1A Q16665 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30884128 0.79 CYP3A4 (0.43) THRBMAOAMAOBCD44MEN1
SCHEMBL135806 0.79 CYP3A4 (0.43) THRBMAOAMAOBCD44MEN1
SCHEMBL11077250 0.75 CYP3A4 (0.40) THRBMAOAMAOBCD44MEN1
Bromide SCHEMBL18245441 0.75 CYP3A4 (0.40) THRBMAOAMAOBCD44MEN1
SCHEMBL11075941 0.75 CYP3A4 (0.40) THRBMAOAMAOBCD44MEN1
Hydrochloric Acid SCHEMBL1198227 0.75 CYP3A4 (0.40) THRBMAOAMAOBCD44MEN1
Hydrochloric Acid SCHEMBL3410713 0.75 CYP3A4 (0.40) THRBMAOAMAOBCD44MEN1
Hydrochloric Acid SCHEMBL11412075 0.75 CYP3A4 (0.40) THRBMAOAMAOBCD44MEN1
SCHEMBL11075931 0.75 CYP3A4 (0.40) THRBMAOAMAOBCD44MEN1
Water SCHEMBL28530113 0.75 CYP3A4 (0.40) THRBMAOAMAOBCD44MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed