SCHEMBL7309211

SCHEMBL7309211

CCc1c(C)nc(N)nc1OC

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.54
TLR8 Q9NR97 12/20 0.53
TLR7 Q9NYK1 8/20 0.53
NUDT1 P36639 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CCNA1 P78396 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26978391 0.87 CCNA2 (0.44) MAPK1TLR8TLR7NUDT1CCNA2
SCHEMBL9287308 0.80 TLR8 (0.55) MAPK1TLR8TLR7NUDT1
SCHEMBL26978000 0.78 MAPK1 (0.46) MAPK1TLR8TLR7NPSR1CCNA2
SCHEMBL30559717 0.78 MAPK1 (0.46) MAPK1TLR8TLR7NPSR1CCNA2
SCHEMBL23264142 0.78 TSHR (0.37) MAPK1TLR8TLR7
SCHEMBL26980485 0.75 TLR8 (0.42) TLR8TLR7CCNA2CDK2CCNA1
SCHEMBL18134204 0.74 CCNA2 (0.44) MAPK1NUDT1NPSR1CCNA2CDK2
SCHEMBL9287284 0.74 CCNA2 (0.44) MAPK1TLR8TLR7NUDT1NPSR1
SCHEMBL31051087 0.72 TLR8 (0.49) MAPK1TLR8TLR7NUDT1
SCHEMBL15434725 0.72 TLR8 (0.49) MAPK1TLR8TLR7NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4588720-A ANXIOLYTIC AGENTS ROUSSEL UCLAF (FR) 1986-05-13 US disclosed
US-4532243-A Imidazo(1,2-a)pyrimidines and their salts useful for treating anxiety ROUSSEL UCLAF (FR) 1985-07-30 US disclosed
EP-0104104-A1 Imidazo(1,2-a)pyrimidines and their salts, process and intermediates for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1984-03-28 EP disclosed