SCHEMBL7309908

SCHEMBL7309908

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CNCC(O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.65
ATM Q13315 1/20 0.62
BCHE P06276 2/20 0.57
BACE1 P56817 5/20 0.56
PSEN1 P49768 3/20 0.54
PSEN2 P49810 3/20 0.54
APH1B Q8WW43 3/20 0.54
NCSTN Q92542 3/20 0.54
APH1A Q96BI3 3/20 0.54
PSENEN Q9NZ42 3/20 0.54
APP P05067 1/20 0.53
CTSS P25774 2/20 0.53
CTSL P07711 1/20 0.53
CTSB P07858 1/20 0.53
CTSK P43235 1/20 0.53
SLC6A11 P48066 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303561 0.96 KLK5 (0.61) KLK5ATMBCHEBACE1PSEN1
SCHEMBL7309398 0.96 KLK5 (0.61) KLK5ATMBCHEBACE1PSEN1
SCHEMBL1236129 0.95 KLK5 (0.61) KLK5ATMBCHEBACE1PSEN1
SCHEMBL1104912 0.95 KLK5 (0.61) KLK5ATMBCHEBACE1PSEN1
SCHEMBL12103325 0.95 KLK5 (0.61) KLK5ATMBCHEBACE1PSEN1
SCHEMBL691498 0.95 KLK5 (0.61) KLK5ATMBCHEBACE1PSEN1
SCHEMBL19261937 0.95 KLK5 (0.61) KLK5ATMBCHEBACE1PSEN1
SCHEMBL8222457 0.95 KLK5 (0.61) KLK5ATMBCHEBACE1PSEN1
SCHEMBL495728 0.94 ATM (0.72) KLK5ATMBCHEBACE1SLC6A11
SCHEMBL4809494 0.94 ATM (0.72) KLK5ATMBCHEBACE1SLC6A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559256-A Aminediol protease inhibitors E. R. SQUIBB & SONS, INC. (US) 1996-09-24 US disclosed
EP-0580402-A2 Aminediol protease inhibitors E.R. SQUIBB & SONS, INC. (US) 1994-01-26 EP disclosed