SCHEMBL7310669

SCHEMBL7310669

O=C(O)OCc1cccnn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.51
CTDSP1 Q9GZU7 1/20 0.51
VNN1 O95497 2/20 0.42
NPC1 O15118 3/20 0.41
LMNA P02545 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
P2RX7 Q99572 1/20 0.41
CYP2C9 P11712 1/20 0.39
NAMPT P43490 1/20 0.39
GABRA1 P14867 2/20 0.37
GABRG2 P18507 2/20 0.37
GABRB3 P28472 2/20 0.37
GABRA5 P31644 2/20 0.37
GABRA3 P34903 2/20 0.37
CES1 P23141 1/20 0.36
NLRP3 Q96P20 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TBXA2R P21731 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25885841 0.78 CYP1A2 (0.53) CYP1A2CTDSP1VNN1NPC1LMNA
SCHEMBL11377704 0.76 SMN1; SMN2 (0.66) CYP1A2NPC1LMNARAB9ASMN1; SMN2
SCHEMBL11318815 0.75 CYP1A2 (0.56) CYP1A2CTDSP1VNN1LMNAP2RX7
Hydrochloric Acid SCHEMBL27803205 0.73 CYP1A2 (0.54) CYP1A2CTDSP1VNN1LMNAP2RX7
SCHEMBL3150298 0.72
Acetic Acid SCHEMBL23877896 0.72 CYP1A2 (0.53) CYP1A2CTDSP1VNN1P2RX7CYP2C9
SCHEMBL31080880 0.72 CYP1A2 (0.53) CYP1A2CTDSP1VNN1P2RX7CYP2C9
SCHEMBL25660463 0.72 CYP1A2 (0.53) CYP1A2CTDSP1VNN1P2RX7CYP2C9
SCHEMBL28021265 0.72 CTDSP1 (0.41) CYP1A2CTDSP1VNN1SMN1; SMN2P2RX7
SCHEMBL6708489 0.72 CTDSP1 (0.41) CYP1A2CTDSP1VNN1P2RX7CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed