SCHEMBL7310856

SCHEMBL7310856

CCC(=O)OC1(c2ccccc2)CCN(CCCC2(c3ccc(Cl)c(Cl)c3)CCCN(C(=O)c3ccccc3)C2)CC1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 16/20 0.73
TACR1 P25103 16/20 0.73
TACR3 P29371 8/20 0.73
CYP3A4 P08684 1/20 0.71
CYP2D6 P10635 1/20 0.71
CYP2C9 P11712 1/20 0.71
CYP2C19 P33261 1/20 0.71
CCR5 P51681 2/20 0.62
DRD3 P35462 1/20 0.55
HRH1 P35367 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8015907 0.99 TACR2 (0.72) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL6450782 0.86 TACR2 (0.71) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL8970867 0.86 TACR2 (0.53) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL6449925 0.85 TACR2 (0.72) TACR2TACR1TACR3CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL6544537 0.85 TACR2 (0.69) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL7090412 0.85 TACR1 (0.79) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL6448486 0.85 TACR1 (0.79) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL6449952 0.85 TACR1 (0.79) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL7305530 0.85 TACR2 (0.74) TACR2TACR1TACR3CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL6543268 0.85 TACR2 (0.71) TACR2TACR1TACR3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673928-A1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists SANOFI (FR) 1995-09-27 EP disclosed