SCHEMBL7312413

SCHEMBL7312413

OC1(c2ccccc2)c2cc(Cl)ccc2-c2ccc(Cl)cc21

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 6/20 0.53
MAP3K14 Q99558 1/20 0.43
P2RX1 P51575 1/20 0.41
P2RX3 P56373 1/20 0.41
P2RX4 Q99571 1/20 0.41
P2RX7 Q99572 1/20 0.41
AKR1A1 P14550 2/20 0.41
AKR1B1 P15121 2/20 0.41
SCN9A Q15858 1/20 0.40
S100A4 P26447 1/20 0.37
MAPT P10636 1/20 0.36
GPR3 P46089 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL824170 0.85 MAP3K14 (0.46) PDK2MAP3K14P2RX1P2RX3P2RX4
SCHEMBL21732768 0.82 PDK2 (0.61) PDK2SCN9A
SCHEMBL19152841 0.79 PDK2 (0.55) PDK2AKR1A1AKR1B1
SCHEMBL26025129 0.78 PDK2 (0.41) PDK2MAP3K14AKR1A1AKR1B1
SCHEMBL25625063 0.78 MAP3K14 (0.41) PDK2MAP3K14P2RX1P2RX3P2RX4
SCHEMBL18167755 0.77 PDK2 (0.56) PDK2MAPT
SCHEMBL7433395 0.77 PDK2 (0.54) PDK2P2RX1P2RX3P2RX4P2RX7
SCHEMBL3038890 0.77 PDK2 (0.53) PDK2P2RX1P2RX3P2RX4P2RX7
SCHEMBL31483494 0.77 PDK2 (0.53) PDK2P2RX1P2RX3P2RX4P2RX7
SCHEMBL23125610 0.76 BCHE (0.45) PDK2MAP3K14P2RX1P2RX3P2RX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6162824-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ALLELIX NEUROSCIENCE INC. 2000-12-19 US disclosed
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO disclosed