SCHEMBL7313607

SCHEMBL7313607

CCc1c(OC)cc(OC)c2c1C(=O)N(CCl)S2(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
ELANE P08246 7/20 0.34
IDO1 P14902 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7288469 0.79 ELANE (0.49) ELANE
SCHEMBL7311933 0.76 ELANE (0.31) ELANE
SCHEMBL7288208 0.71 ELANE (0.39) ELANE
SCHEMBL7305964 0.70 ELANE (0.77) ELANE
SCHEMBL7288666 0.69 ELANE (0.58) ELANE
SCHEMBL7290646 0.69 ELANE (0.55) ELANE
SCHEMBL7304815 0.69 PDE3B (0.37) PDE3BPDE3AIDO1
SCHEMBL7278505 0.68 ELANE (0.53) ELANE
SCHEMBL7304861 0.67 ELANE (0.37) ELANE
SCHEMBL7278649 0.66 ELANE (0.61) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874432-A Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof SANOFI (FR) 1999-02-23 US disclosed
US-5650422-A TREATMENT OF EMPHYSEMA, ARTHRITIS OR PANCREATITIS SANOFI (FR) 1997-07-22 US disclosed
US-5596012-A Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof STERLING WINTHROP INC. (US) 1997-01-21 US disclosed
US-5371074-A Use of saccharin derivatives as proteolytic enzyme inhibitors STERLING WINTHROP INC. (US) 1994-12-06 US disclosed
US-5236917-A Respiratory system disorders, antiarthritic agents STERLING WINTHROP INC. (US) 1993-08-17 US disclosed
EP-0542372-A1 2-Substituted saccharin derivative proteolytic enzyme inhibitors STERLING WINTHROP INC. (US) 1993-05-19 EP disclosed