SCHEMBL7313783

SCHEMBL7313783

CC(C)(C)c1ccn(-c2ccc(C(=O)N3Cc4cccnc4Nc4ccccc43)c(C(F)(F)F)c2)n1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 9/20 0.83
AVPR1A P37288 3/20 0.83
IDH1 O75874 11/20 0.47
OXTR P30559 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6617257 0.94 AVPR2 (0.84) AVPR2AVPR1AIDH1
SCHEMBL6614886 0.91 AVPR2 (1.00) AVPR2AVPR1AIDH1OXTR
SCHEMBL6615073 0.86 AVPR2 (0.78) AVPR2AVPR1AIDH1OXTR
SCHEMBL7318297 0.82 AVPR2 (1.00) AVPR2AVPR1AIDH1
SCHEMBL6616064 0.81 AVPR2 (0.71) AVPR2AVPR1AIDH1
SCHEMBL7312662 0.80 AVPR2 (1.00) AVPR2AVPR1AIDH1OXTR
SCHEMBL7312434 0.80 AVPR2 (0.54) AVPR2AVPR1AIDH1
SCHEMBL6615031 0.78 AVPR2 (0.52) AVPR2AVPR1AIDH1
SCHEMBL6616836 0.78 AVPR2 (1.00) AVPR2AVPR1AIDH1OXTR
SCHEMBL6615751 0.78 AVPR2 (1.00) AVPR2AVPR1AIDH1OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1149096-B1 TRICYCLIC PYRIDINE N-OXIDES VASOPRESSIN AGONISTS WYETH CORP (US) 2002-12-18 EP disclosed
US-6235900-B1 Tricyclic pyridine N-oxides vasopressin agonists AMERICAN HOME PRODUCTS CORPORATION 2001-05-22 US disclosed