SCHEMBL7314948

SCHEMBL7314948

CCn1c(=O)c2c(nc(C=Cc3cccc(Cl)c3)n2C)n(CC)c1=O

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.74
MAOB P27338 2/20 0.70
ADORA2B P29275 2/20 0.70
CYP1A2 P05177 1/20 0.70
CYP2D6 P10635 1/20 0.70
HIF1A Q16665 1/20 0.70
HSD17B10 Q99714 1/20 0.70
KDM4E B2RXH2 1/20 0.70
ALDH1A1 P00352 1/20 0.70
GLA P06280 1/20 0.70
HPGD P15428 1/20 0.70
AHR P35869 1/20 0.70
BLM P54132 1/20 0.70
PMP22 Q01453 1/20 0.70
HTR1A P08908 1/20 0.67
ADORA3 P0DMS8 1/20 0.67
CYP2C9 P11712 1/20 0.67
PDE4A P27815 1/20 0.67
ADORA1 P30542 1/20 0.67
PDE4D Q08499 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7314940 1.00 ADORA2A (0.74) ADORA2AMAOBADORA2BCYP1A2CYP2D6
SCHEMBL5142398 0.91 ADORA2A (0.70) ADORA2AMAOBADORA2BCYP1A2CYP2D6
SCHEMBL5142395 0.91 ADORA2A (0.70) ADORA2AMAOBADORA2BCYP1A2CYP2D6
SCHEMBL7314398 0.88 ADORA2A (0.76) ADORA2AMAOBADORA2BHTR1AADORA3
SCHEMBL7282865 0.88 ADORA2A (0.73) ADORA2AMAOBADORA2BHTR1AADORA3
SCHEMBL7282856 0.88 ADORA2A (0.73) ADORA2AMAOBADORA2BHTR1AADORA3
SCHEMBL7541313 0.88 ADORA2A (0.73) ADORA2AMAOBADORA2BHTR1AADORA3
SCHEMBL7541320 0.88 ADORA2A (0.73) ADORA2AMAOBADORA2BHTR1AADORA3
SCHEMBL7314391 0.88 ADORA2A (0.76) ADORA2AMAOBADORA2BHTR1AADORA3
SCHEMBL7279473 0.86 ADORA2A (0.73) ADORA2AMAOBADORA2BGLAHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628311-B1 Xanthine-Derivatives as Antidepressants KYOWA HAKKO KOGYO KK (JP) 2002-04-24 EP disclosed
US-5587378-A ADMINISTERING A SUBSTITUTED XANTHINE COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-12-24 US disclosed
US-5543415-A ADMINISTERING A XANTHINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-08-06 US disclosed
US-5484920-A XANTHINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-01-16 US disclosed
EP-0628311-A1 ANTIDEPRESSANT KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-12-14 EP disclosed
EP-0590919-A1 Therapeutic agents for parkinson's disease KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-04-06 EP disclosed