SCHEMBL7318610

SCHEMBL7318610

N#Cc1cn2cc(Br)nc(N3CCOCC3)c2n1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.43
ALDH1A1 P00352 7/20 0.40
HPGD P15428 4/20 0.40
KHK P50053 1/20 0.40
HTR2C P28335 1/20 0.39
MAPK1 P28482 2/20 0.38
KDM4E B2RXH2 6/20 0.38
HSD17B10 Q99714 3/20 0.38
TSHR P16473 1/20 0.37
RXFP1 Q9HBX9 2/20 0.37
CLK1 P49759 1/20 0.37
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10092233 0.79 PIK3CA (0.55) ALDH1A1HPGDKHKHTR2CMAPK1
SCHEMBL2448071 0.77 PIK3CA (0.41) ALDH1A1HPGDHTR2CMAPK1KDM4E
SCHEMBL26072464 0.77 PIK3R1 (0.46) HTR2CPIK3R1PIK3CA
SCHEMBL5561919 0.76 HTR2C (0.39) ALDH1A1HTR2CMAPK1TSHRPIK3R1
SCHEMBL5560455 0.76 PIK3CA (0.58) HTR2CPIK3R1PIK3CA
SCHEMBL10092212 0.76 PIK3R1 (0.45) HTR2CPIK3R1PIK3CA
SCHEMBL13896920 0.76 PIK3CA (0.45) HTR2CPIK3R1PIK3CA
SCHEMBL26072359 0.75 PIK3CA (0.50) HTR2CRXFP1PIK3R1PIK3CAPOLB
SCHEMBL5560237 0.74 PIK3CA (0.64) HTR2CKDM4EHSD17B10PIK3R1PIK3CA
SCHEMBL10092229 0.74 PIK3CA (0.49) HTR2CPIK3R1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5028605-A Antispasmodic, bronchodilators, uterine relaxants, cardiac analeptics, neurosedatives L'UNIVERSITE DE MONTPELLIER I (FR) 1991-07-02 US disclosed
EP-0348392-A1 8-ALKYLAMINOIMIDAZO[1,2-A]PYRAZINES AND DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY Université Montpellier I (FR) 1990-01-03 EP disclosed
WO-1988004298-A1 8-ALKYLAMINOIMIDAZO[1,2-A]PYRAZINES AND DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1988-06-16 WO disclosed