SCHEMBL7322970

SCHEMBL7322970

CCOC(=O)c1ccccc1/C=C/c1ccc2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.51
CAPN1 P07384 2/20 0.50
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
CNR2 P34972 1/20 0.49
CDC25B P30305 2/20 0.48
PTGS1 P23219 1/20 0.47
ALDH1A1 P00352 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NQO2 P16083 2/20 0.44
GAA P10253 1/20 0.44
RELA Q04206 1/20 0.44
PPARA Q07869 1/20 0.44
PTGS2 P35354 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7322975 1.00 TSHR (0.51) TSHRCAPN1CTSLCTSBCNR2
SCHEMBL7790064 0.83 TSHR (0.61) TSHRCDC25BALDH1A1HSD17B10
SCHEMBL27533745 0.83 TSHR (0.61) TSHRCDC25BALDH1A1HSD17B10
SCHEMBL7324455 0.82 CYP1A1 (0.58) TSHRCAPN1ALDH1A1
SCHEMBL7324446 0.82 CYP1A1 (0.58) TSHRCAPN1ALDH1A1
Hydrochloric Acid SCHEMBL6800822 0.81 TSHR (0.44) TSHRCNR2CDC25BPTGS1ALDH1A1
Dimethylamine SCHEMBL1335350 0.80 TSHR (0.53) TSHRCDC25BALDH1A1HSD17B10
SCHEMBL9000589 0.79 TSHR (0.59) TSHRCDC25BALDH1A1HSD17B10
SCHEMBL9000587 0.79 TSHR (0.59) TSHRCDC25BALDH1A1HSD17B10
SCHEMBL7322163 0.79 GRIK1 (0.59) CAPN1CTSLCTSBPTGS1RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
US-6103720-A ENZYME INHIBITORS; ANTIICHEMIC AND -TUMOR AGENTS; STROKES; ALZEIMER'S DISEASE BASF AKTIENGESELLSCHAFT (DE) 2000-08-15 US disclosed
CN-1245486-A Ketobenzamides as calpain inhibitors BASF AG (DE) 2000-02-23 CN disclosed
CN-1238761-A benzamide aldehydes and their use as cysteine protease inhibitors BASF AG (DE) 1999-12-15 CN disclosed