SCHEMBL7325474

SCHEMBL7325474

[CH2]CN1CCC(C(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.68
HTR2C P28335 2/20 0.68
HTR7 P34969 2/20 0.68
HTR6 P50406 2/20 0.68
HSD11B1 P28845 1/20 0.63
LMNA P02545 2/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
HTT P42858 1/20 0.63
KDM4E B2RXH2 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10928970 0.88 HTR2A (0.72) HTR2AHTR2CHTR7HTR6HSD11B1
SCHEMBL14318600 0.87 HTR2A (0.81) HTR2AHTR2CHTR7HTR6HSD11B1
SCHEMBL11107232 0.84 HTR2A (0.68) HTR2AHTR2CHTR7HTR6HSD11B1
SCHEMBL9879782 0.84 HTR2A (0.63) HTR2AHTR2CHTR7HTR6HSD11B1
SCHEMBL8714691 0.83 HTR2A (0.74) HTR2AHTR2CHTR7HTR6HSD11B1
SCHEMBL9499649 0.83 SMN1; SMN2 (0.69) HTR2AHTR2CHTR7HTR6HSD11B1
SCHEMBL14636954 0.83 SMN1; SMN2 (0.69) HTR2AHTR2CHTR7HTR6HSD11B1
SCHEMBL14282300 0.83 HTR2A (0.66) HTR2AHTR2CHTR7HTR6HSD11B1
SCHEMBL10928975 0.82 HTR2A (0.72) HTR2AHTR2CHTR7HTR6HSD11B1
Hydrochloric Acid SCHEMBL9502312 0.82 SMN1; SMN2 (0.67) HTR2AHTR2CHTR7HTR6HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0377528-B1 Piperidines, process for their preparation and pharmaceutical compounds containing them LIPHA (FR) 1993-12-08 EP claimed
US-5001134-A Piperidines, processes of preparation and medications containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1991-03-19 US claimed
US-4032642-A SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1977-06-28 US claimed
US-3956296-A ANTIINFLAMMATORY, SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1976-05-11 US claimed
WO-2000024715-A1 PIPERIDINE COMPOUNDS AND THEIR USE IN THE POPULATION CONTROL OF RODENTS AND OTHER VERTEBRATE PESTS ALMIRALL PRODESFARMA, S.A. (ES) 2000-05-04 WO disclosed
US-5001134-A Piperidines, processes of preparation and medications containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1991-03-19 US disclosed
US-5001134-A Piperidines, processes of preparation and medications containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1991-03-19 US disclosed
EP-0377528-A1 Piperidines, process for their preparation and pharmaceutical compounds containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1990-07-11 EP disclosed
US-4032642-A SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1977-06-28 US disclosed
US-4032642-A SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1977-06-28 US disclosed
US-3956296-A ANTIINFLAMMATORY, SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1976-05-11 US disclosed
US-3956296-A ANTIINFLAMMATORY, SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1976-05-11 US disclosed