SCHEMBL7326146

SCHEMBL7326146

CCOC(=O)CN(C(=O)[C@H](CC(=O)OC(C)(C)C)NS(=O)(=O)c1ccc2ccccc2c1)C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.45
ACACB O00763 1/20 0.43
F2 P00734 6/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PLG P00747 1/20 0.41
KAT6A Q92794 1/20 0.40
PLAU P00749 1/20 0.38
PLAT P00750 1/20 0.38
BACE1 P56817 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8721707 0.91 GAA (0.47) GAAF2ALDH1A1MEN1KMT2A
SCHEMBL8716864 0.89 GAA (0.45) GAAACACBF2ALDH1A1MEN1
SCHEMBL7302360 0.86 ACACB (0.45) GAAACACBF2PLGPLAU
SCHEMBL7327272 0.86 GAA (0.42) GAAACACBF2ALDH1A1MEN1
SCHEMBL7334523 0.86 GAA (0.42) GAAACACBF2ALDH1A1MEN1
SCHEMBL8947835 0.85 GAA (0.42) GAAACACBF2ALDH1A1MEN1
SCHEMBL7332989 0.85 F2 (0.47) ACACBF2PLGPLAT
SCHEMBL7332615 0.85 F2 (0.49) F2PLGPLAT
SCHEMBL8719583 0.84 F2 (0.48) F2PLGPLAT
SCHEMBL7395628 0.83 GAA (0.48) GAAACACBF2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559046-B1 N-amidinopiperidinyl(3/4)- or N-amidino-1,4-Oxazinyl(2)-substituted sulfonamides, process for their preparation and use as thrombin inhibitors HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
EP-0559046-A1 N-amidinopiperidinyl(3/4)- or N-amidino-1,4-Oxazinyl(2)-substituted sulfonamides, process for their preparation and use as thrombin inhibitors F.HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT (CH) 1993-09-08 EP disclosed