SCHEMBL7327110

SCHEMBL7327110

CC(C)CCC(N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)O)C(=O)OCc1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACE P12821 15/20 0.74
LMNA P02545 2/20 0.74
SMN1; SMN2 Q16637 1/20 0.68
ABCB11 O95342 1/20 0.52
ACE2 Q9BYF1 4/20 0.50
PREP P48147 2/20 0.50
MEN1 O00255 1/20 0.50
USP2 O75604 1/20 0.50
KMT2A Q03164 1/20 0.50
CYP3A4 P08684 1/20 0.50
ALOX15 P16050 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7321931 0.92 ACE (0.87) ACELMNASMN1; SMN2ABCB11MEN1
SCHEMBL6418176 0.92 ACE (0.87) ACELMNASMN1; SMN2ABCB11MEN1
SCHEMBL7320701 0.88 ACE (0.68) ACELMNASMN1; SMN2ACE2
SCHEMBL7359927 0.88 ACE (0.67) ACELMNASMN1; SMN2ACE2PREP
SCHEMBL7329937 0.88 ACE (0.67) ACELMNASMN1; SMN2ACE2PREP
SCHEMBL14282793 0.85 ACE (0.76) ACELMNASMN1; SMN2ABCB11MEN1
Enalapril SCHEMBL8433334 0.85 ACE (1.00) ACELMNASMN1; SMN2ABCB11MEN1
Enalapril SCHEMBL6159149 0.85 ACE (1.00) ACELMNASMN1; SMN2ABCB11MEN1
Enalapril SCHEMBL474012 0.85 ACE (1.00) ACELMNASMN1; SMN2ABCB11MEN1
Enalapril SCHEMBL97 0.85 ACE (1.00) ACELMNASMN1; SMN2ABCB11MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4472380-A CARBOXYALKYL DIPEPTIDE DERIVATIVES MERCK & CO., INC. (US) 1984-09-18 US disclosed
US-4374829-A Aminoacid derivatives as antihypertensives MERCK & CO., INC. (US) 1983-02-22 US disclosed
EP-0012401-A1 Carboxyalkyl dipeptide derivatives, process for preparing them and pharmaceutical composition containing them MERCK & CO. INC. (US) 1980-06-25 EP disclosed