SCHEMBL7327375

SCHEMBL7327375

CCCCCCCCCCN(C)CCCC(C#N)(c1ccc(OC)c(OC)c1)C(C)C

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 9/20 0.76
CYP3A4 P08684 7/20 0.76
ABCC1 P33527 4/20 0.76
KCNH2 Q12809 3/20 0.76
TSHR P16473 3/20 0.76
LMNA P02545 3/20 0.76
MEN1 O00255 3/20 0.76
KMT2A Q03164 3/20 0.76
CYP2C19 P33261 2/20 0.76
ABCB11 O95342 2/20 0.76
CACNA1F O60840 2/20 0.76
HTR1A P08908 2/20 0.76
ADRA2A P08913 2/20 0.76
DRD2 P14416 2/20 0.76
ADRA2C P18825 2/20 0.76
HTR2A P28223 2/20 0.76
HTR2C P28335 2/20 0.76
SLC6A4 P31645 2/20 0.76
DRD3 P35462 2/20 0.76
SCN1A P35498 2/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7334533 1.00 ABCB1 (0.76) ABCB1CYP3A4ABCC1KCNH2TSHR
SCHEMBL6390800 0.99 ABCB1 (0.77) ABCB1CYP3A4ABCC1KCNH2TSHR
SCHEMBL7623326 0.90 ABCB1 (0.74) ABCB1CYP3A4ABCC1KCNH2TSHR
SCHEMBL7628055 0.89 ABCB1 (0.75) ABCB1CYP3A4ABCC1KCNH2TSHR
Nexopamil SCHEMBL1980872 0.88 ABCB1 (0.70) ABCB1CYP3A4ABCC1KCNH2TSHR
Nexopamil SCHEMBL7265602 0.88 ABCB1 (0.70) ABCB1CYP3A4ABCC1KCNH2TSHR
SCHEMBL7272996 0.88 ABCB1 (0.70) ABCB1CYP3A4ABCC1KCNH2TSHR
SCHEMBL6386436 0.88 ABCB1 (0.77) ABCB1CYP3A4ABCC1KCNH2TSHR
SCHEMBL6387767 0.88 ABCB1 (0.77) ABCB1CYP3A4ABCC1KCNH2TSHR
SCHEMBL7273704 0.88 ABCB1 (0.70) ABCB1CYP3A4ABCC1KCNH2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0434093-A1 Omega-amino-alpha-phenylalkano-nitrile derivatives G.D. Searle & Co. (US) 1991-06-26 EP claimed
US-5643947-A CALCIUM CHANNEL BLOCKER G. D. SEARLE & CO. (US) 1997-07-01 US disclosed